Tasimelteon (ab272096)
Key features and details
- Dual-acting metatonin MT1/MT2 receptor agonist
- CAS Number: 609799-22-6
- Soluble in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
製品の概要
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製品名
Tasimelteon -
製品の詳細
Dual-acting metatonin MT1/MT2 receptor agonist -
生理活性の詳細
Dual-acting metatonin MT1/MT2 receptor agonist. Binds MT2 receptor with greater affinity (Ki = 0.0692 - 0.17 nM, depending on cell type) than the MT1 receptor (Ki = 0.304-0.35 nM). No significant affinity towards a panel of 160 pharmacologically important receptors and enzymes. Resets the circadian master clock. Used in the treatment of non-24 hour sleep-wake disorder.
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CAS 番号
609799-22-6 -
構造式
製品の特性
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体系名
N-[[(1R,2R)-2-(2,3-Dihydro-4-benzofuranyl)cyclopropyl]methyl]propanamide -
分子量
245.32 -
分子式
C15H19NO2 -
PubChem 登録番号
10220503 -
保存方法
Shipped at Room Temperature. Store at +4°C. -
溶解性
Soluble in DMSO to 100 mM -
使用に関する注意
Refer to SDS for further information
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES 線形表記
CCC(=O)NC[C@@H]1C[C@H]1C2=C3CCOC3=CC=C2 -
由来
Synthetic
画像
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Chemical Structure - Tasimelteon (ab272096)
Chemical structure of Tasimelteon, 609799-22-6
プロトコール
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
データシートおよび資料
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SDS download
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Datasheet download
参考文献 (0)
ab272096 は論文での使用が確認できていません。