SM64, beta1 adrenoceptor antagonist (ab144659)
Key features and details
- Highly selective β1 adrenoceptor antagonist and partial agonist
- CAS Number:
- Purity: > 97%
- Soluble in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
製品の概要
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製品名
SM64, beta1 adrenoceptor antagonist -
製品の詳細
Highly selective β1 adrenoceptor antagonist and partial agonist -
生理活性の詳細
Highly selective β1 adrenoceptor antagonist (log KD = -7.5 for β1 and incomplete binding inhibition for β2). Exhibits β1-partial agonist activity (log EC50 = -8; 34% isoprenalinie maximum). Active in vitro and in vivo.
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精製度
> 97% -
構造式
製品の特性
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体系名
1-[2-[[3-[4-[2-(Cyclopropylmethoxy)ethoxy]phenoxy]-2-hydroxypropyl]amino]ethyl]-3-(4-hydroxyphenyl)urea -
分子量
459.54 -
分子式
C24H33N3O6 -
保存方法
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
溶解性
Soluble in DMSO to 100 mM -
使用に関する注意
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES 線形表記
Oc1ccc(cc1)NC(=O)NCCNCC(O)COc3ccc(OCCOCC2CC2)cc3 -
由来
Synthetic
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研究分野
画像
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Chemical Structure - SM64, beta1 adrenoceptor antagonist (ab144659)2D chemical structure image of ab144659, SM64, beta1adrenoceptor antagonist
プロトコール
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
参考文献 (0)
ab144659 は論文での使用が確認できていません。
