CTAP, mu opioid antagonist (ab120680)
Key features and details
- Potent, selective μ opioid antagonist
- CAS Number: 103429-32-9
- Soluble in water
- Form / State: Solid
- Source: Synthetic
製品の概要
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製品名
CTAP, mu opioid antagonist -
製品の詳細
Potent, selective μ opioid antagonist -
生理活性の詳細
Potent and selective μ opioid receptor antagonist (1200-fold more selective vs. δ receptor). Blood-brain barrier permeable and active in vivo. Antagonizes antinociceptive effect.
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CAS 番号
103429-32-9 -
構造式
製品の特性
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分子量
1104.31 -
分子式
C51H69N13O11S2 -
配列
FCYWRTXT (Modifications: C-terminal amide; X-7 = Pen; Phe-1 = D-Phr; Trp-4 = D-Trp; Disulfide bonds: 2-7) -
保存方法
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
溶解性
Soluble in water -
使用に関する注意
This product is supplied in one (or more) pack size which is freeze dried. Therefore the contents may not be readily visible, as they can coat the bottom or walls of the vial. Please see our FAQs and information page for more details on handling.
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one week. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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由来
Synthetic
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研究分野
プロトコール
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
参考文献 (1)
ab120680 は 1 報の論文で使用されています。
- Furukawa A et al. Endothelin Signaling Contributes to Modulation of Nociception in Early-stage Tongue Cancer in Rats. Anesthesiology 128:1207-1219 (2018). PubMed: 29461271