製品の概要

  • 製品名Varenicline tartrate
  • 製品の詳細
    Orally active partial agonist at α4β2 nicotinic receptors
  • 生理活性の詳細High affinity, subtype-selective partial agonist at α4β2 nicotinic receptors. (Ki values are 0.06 (α4β2), 240 (α3β4), 322 (α7) and 3540 nM (α1βγδ)). Full agonist at α7 receptors. Orally active.
  • 精製度> 99%

製品の特性

  • 体系名7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino[2,3-h][3]benzazepine tartrate
  • 分子量361.37
  • 構造式Chemical Structure
  • 分子式C13H13N3.C4H6O6
  • CAS 番号375815-87-5
  • 保存方法Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months.
  • 溶解性Soluble in water to 100 mM
  • 使用に関する注意

    Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.

    Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.

  • 由来

    Synthetic

  • 研究分野

    Varenicline tartrate (ab120539) 使用論文

    This product has been referenced in:

    See all 4 Publications for this product

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